SCHEMBL257625

SCHEMBL257625

COc1ccc(Oc2ccc(C)cc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.83
LTA4H P09960 2/20 0.64
RELA Q04206 1/20 0.62
CA1 P00915 2/20 0.61
CA2 P00918 2/20 0.61
CA7 P43166 2/20 0.61
CA9 Q16790 2/20 0.61
CA12 O43570 1/20 0.61
CA14 Q9ULX7 1/20 0.61
TEAD4 Q15561 1/20 0.61
ALDH1A1 P00352 3/20 0.58
TDP1 Q9NUW8 2/20 0.58
MAPT P10636 2/20 0.58
POLB P06746 1/20 0.58
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
PARP10 Q53GL7 1/20 0.50
AR P10275 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12277315 1.00 ACHE (0.83) ACHELTA4HRELACA1CA2
SCHEMBL12335539 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL14826485 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL12770837 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL10044180 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL12276818 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL12770835 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL12334794 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL12761860 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2
SCHEMBL18708707 0.93 ACHE (0.71) ACHELTA4HRELACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 237 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059107-A1 IKZF2 AND CK1-ALPHA DEGRADING COMPOUNDS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2024-03-21 WO disclosed
US-20240019738-A1 DISPLAY DEVICE AND MANUFACTURING METHOD THEREOF JAPAN DISPLAY INC. (JP) 2024-01-18 US disclosed
WO-2023190767-A1 POLYETHER ETHER KETONE DECOMPOSITION METHOD AND NOVEL SUBSTANCE USING STARTING MATERIAL THAT IS DECOMPOSITION PRODUCT OBTAINED BY THIS DECOMPOSITION METHOD 国立研究開発法人産業技術総合研究所 2023-10-05 WO disclosed
EP-3326715-B1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE CE PHARM CO LTD (CN) 2021-09-15 EP disclosed
WO-2021156636-A1 TRIAZOLE DERIVATIVES WITH ANTIFUNGAL ACTIVITY KING'S COLLEGE LONDON (GB) 2021-08-12 WO disclosed
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed
WO-2020121577-A1 EPOXY COMPOUND JNC株式会社 2020-06-18 WO disclosed
US-10465046-B2 Polyarylether ketone imide adhesives THE BOEING COMPANY (US) 2019-11-05 US disclosed
WO-2019173507-A1 ANTIBACTERIAL AGENTS : ARYLALKYLCARBOXAMIDO PHLOROGLUCINOLS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2019-09-12 WO disclosed
WO-2019142927-A1 LIQUID CRYSTAL ALIGNING AGENT, LIQUID CRYSTAL ALIGNMENT FILM, AND LIQUID CRYSTAL DISPLAY ELEMENT USING SAME 日産化学株式会社 2019-07-25 WO disclosed
EP-0603889-A2 Process for the preparation of lactic acid polyesters MITSUI TOATSU CHEMICALS, Inc. (JP) 1994-06-29 EP disclosed
US-5310865-A Polyhydroxycarboxylic acid and preparation process thereof MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-05-10 US disclosed
EP-0572675-A1 POLYHYDROXY CARBOXYLIC ACID AND PRODUCTION THEREOF MITSUI TOATSU CHEMICALS, Inc. (JP) 1993-12-08 EP disclosed
WO-1993013067-A1 4-SUBSTITUTED PIPERIDINECARBOXYLIC ACID ESTERS: INHIBITION OF CHOLESTEROL ABSORPTION AMERICAN HOME PRODUCTS CORPORATION (US) 1993-07-08 WO disclosed
US-5169844-A Enzyme inhibitor, anticholesterol and antilipemic agent AMERICAN HOME PRODUCTS CORPORATION (US) 1992-12-08 US disclosed
EP-0428385-A1 Cholesterol ester hydrolase inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1991-05-22 EP disclosed
US-4391995-A 4-Phenoxy-phenoxy-alkane-carboxylic acid derivatives and process for their manufacture HOECHST AKTIENGESELLSCHAFT (DE) 1983-07-05 US disclosed
US-4301295-A ANTILIPEMIC AND ANTICHOLESTEROL AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1981-11-17 US disclosed
US-4238626-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1980-12-09 US disclosed
US-4113782-A CATALYTIC OXIDATION AGENCY OF INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 1978-09-12 US disclosed