SCHEMBL25768632

SCHEMBL25768632

Cc1cc(-c2ccccc2)nc2ccc(Oc3c(Cl)cc(-n4nc(C#N)c(=O)[nH]c4=O)cc3Br)cc12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 16/20 0.44
THRA P10827 15/20 0.44
CYP2C8 P10632 1/20 0.44
CYP2C9 P11712 1/20 0.44
BCAT1 P54687 1/20 0.34
NPC1 O15118 2/20 0.34
MAPT P10636 2/20 0.34
HTT P42858 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
OPRK1 P41145 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31300999 1.00 THRB (0.44) THRBTHRACYP2C8CYP2C9BCAT1
SCHEMBL30460702 0.95 THRB (0.49) THRBTHRACYP2C8CYP2C9BCAT1
SCHEMBL25291901 0.95 THRB (0.49) THRBTHRACYP2C8CYP2C9BCAT1
SCHEMBL30460745 0.93 THRB (0.37) THRBTHRACYP2C8CYP2C9SMN1; SMN2
SCHEMBL25768247 0.91 THRA (0.48) THRBTHRACYP2C8CYP2C9NPC1
SCHEMBL30460697 0.91 THRA (0.48) THRBTHRACYP2C8CYP2C9NPC1
SCHEMBL25768246 0.89 THRA (0.49) THRBTHRACYP2C8CYP2C9NPC1
SCHEMBL30460753 0.89 THRA (0.49) THRBTHRACYP2C8CYP2C9NPC1
SCHEMBL31301011 0.89 THRB (0.39) THRBTHRACYP2C8CYP2C9SMN1; SMN2
SCHEMBL30460704 0.88 THRB (0.42) THRBTHRACYP2C9MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125716-A1 CLASS OF QUINOLINE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国科学院上海药物研究所 2023-07-06 WO disclosed