SCHEMBL25791708

SCHEMBL25791708

COc1cnc2c(C)cnn2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR2 P37173 3/20 0.51
ACVR2A P27037 1/20 0.51
KDR P35968 12/20 0.45
FLT1 P17948 3/20 0.45
FLT4 P35916 3/20 0.45
PLK4 O00444 1/20 0.45
AURKA O14965 1/20 0.45
DYRK3 O43781 1/20 0.45
MAP4K4 O95819 1/20 0.45
NTRK1 P04629 1/20 0.45
INSR P06213 1/20 0.45
CDK1 P06493 1/20 0.45
FGFR1 P11362 1/20 0.45
CDK2 P24941 1/20 0.45
MARK3 P27448 1/20 0.45
FLT3 P36888 1/20 0.45
CLK2 P49760 1/20 0.45
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
IRAK1 P51617 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13822288 0.80 KDR (0.68) TGFBR2ACVR2AKDRFLT1FLT4
SCHEMBL22834516 0.80 TGFBR2 (0.50) TGFBR2ACVR2AKDRFLT1FLT4
SCHEMBL15308505 0.76 PDE2A (0.41) TGFBR2ACVR2AKDRFLT1FLT4
SCHEMBL17052954 0.76 TGFBR2 (0.47) TGFBR2ACVR2AKDRFLT1FLT4
SCHEMBL359148 0.76 HSD11B1 (0.52) TGFBR2ACVR2AKDRFLT1FLT4
SCHEMBL22834740 0.75 HSD11B1 (0.43) TGFBR2ACVR2AKDRFLT1FLT4
SCHEMBL28979830 0.73 KDR (0.33) KDRFLT1FLT4PLK4AURKA
SCHEMBL25791703 0.73 KDR (0.36) KDRFLT1FLT4PLK4AURKA
SCHEMBL13960990 0.73 KDR (0.37) KDRFLT1FLT4PLK4AURKA
SCHEMBL23728470 0.73 ALDH1A1 (0.54) HSD11B1PDE2AIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023130054-A2 HETEROARYL COMPOUNDS AS INHIBITORS OF IRAK4, COMPOSITIONS AND APPLICATIONS THEREOF ACCRO BIOSCIENCE (HK) LIMITED (CN) 2023-07-06 WO disclosed