SCHEMBL257938

SCHEMBL257938

CC1(C)OC(c2cccc3cc[nH]c23)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.42
NR3C1 P04150 14/20 0.40
PGR P06401 5/20 0.38
KEAP1 Q14145 1/20 0.38
NR3C2 P08235 3/20 0.37
AR P10275 3/20 0.37
PDPK1 O15530 1/20 0.37
BCHE P06276 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488782 0.73 AHR (0.42) AHRNR3C1PGRBCHE
SCHEMBL15499617 0.71 ATM (0.37) AHRNR3C1PGRNR3C2AR
SCHEMBL7864768 0.69 AHR (0.48) AHRNR3C1PGRKEAP1NR3C2
SCHEMBL21149281 0.67 AHR (0.46) AHRNR3C1PGRKEAP1NR3C2
SCHEMBL29469161 0.67 AHR (0.42) AHRNR3C1PGRKEAP1NR3C2
SCHEMBL2028185 0.67 AHR (0.42) AHRNR3C1PGRKEAP1NR3C2
SCHEMBL9946124 0.65 NPSR1 (0.41)
SCHEMBL31637123 0.65 CYP3A4 (0.48)
SCHEMBL9688985 0.65 AHR (0.47) AHRNR3C1PGRKEAP1NR3C2
SCHEMBL4882951 0.64 HTR2C (0.49) AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed