SCHEMBL25795129

SCHEMBL25795129

Cc1cc(-c2cn[nH]c2)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.46
NPBWR1 P48145 2/20 0.44
KCNH2 Q12809 2/20 0.39
AKT1 P31749 1/20 0.39
AKT2 P31751 1/20 0.39
FDPS P14324 1/20 0.39
EPHB4 P54760 1/20 0.39
LMNA P02545 1/20 0.38
APEX1 P27695 1/20 0.38
PMP22 Q01453 1/20 0.38
PIM1 P11309 2/20 0.38
PIM3 Q86V86 2/20 0.38
PIM2 Q9P1W9 2/20 0.38
PDE4B Q07343 2/20 0.38
CNR1 P21554 1/20 0.38
IDO1 P14902 1/20 0.36
IKBKB O14920 1/20 0.36
RET P07949 1/20 0.36
LRRK2 Q5S007 1/20 0.36
ERN1 O75460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27476106 0.82 KCNH2 (0.52) KCNH2AKT1AKT2FDPSLMNA
SCHEMBL25798414 0.80 NPBWR1 (0.44) NPBWR1KCNH2AKT1AKT2FDPS
SCHEMBL30549950 0.80 NPBWR1 (0.44) NPBWR1KCNH2AKT1AKT2FDPS
SCHEMBL20040983 0.80 NPBWR1 (0.44) NPBWR1KCNH2AKT1AKT2FDPS
SCHEMBL16054951 0.80 NPBWR1 (0.44) NPBWR1KCNH2AKT1AKT2FDPS
SCHEMBL12583213 0.78 NOTUM (0.50) NOTUMIKBKB
SCHEMBL26375464 0.78 NOTUM (0.50) NOTUMIDO1IKBKB
SCHEMBL28182653 0.76 KCNH2 (0.54) KCNH2AKT1AKT2FDPSLMNA
SCHEMBL13949153 0.76 NOTUM (0.49) NOTUMIDO1IKBKB
SCHEMBL2996698 0.75 RXRA (0.50) NPBWR1KCNH2AKT1AKT2FDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109912-A1 3, 4-DIHYDROISOQUINOLIN-1 (2H) -ONES DERIVATIVES AS STING ANTAGONISTS AND THE USE THEREOF BEIGENE, LTD. (KY) 2023-06-22 WO disclosed