SCHEMBL25798970

SCHEMBL25798970

Cc1cc(N[C@@H]2C[C@@H](F)CN(C(C)C)C2)nnc1-c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 3/20 0.46
IL1B P01584 10/20 0.36
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
MAPK14 Q16539 5/20 0.34
PIM1 P11309 1/20 0.33
TNF P01375 1/20 0.33
CSNK1D P48730 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25798600 0.91 IL1B (0.41) NLRP3IL1BTNF
SCHEMBL25798590 0.89 IL1B (0.44) NLRP3IL1BPIM1TNF
SCHEMBL25798535 0.86 NLRP3 (0.55) NLRP3IL1BMAPK14PIM1TNF
SCHEMBL25798527 0.83 NLRP3 (0.60) NLRP3IL1BMAPK14
SCHEMBL25798595 0.83 NLRP3 (0.46) NLRP3IL1BMAPK14
SCHEMBL25798531 0.74 IL1B (0.58) NLRP3IL1BTNF
SCHEMBL25797816 0.74 IL1B (0.58) NLRP3IL1BTNF
SCHEMBL25798896 0.74 NLRP3 (0.68) NLRP3IL1BMAPK14
SCHEMBL25798598 0.74 NLRP3 (0.42) NLRP3IL1B
SCHEMBL25798449 0.73 NLRP3 (0.53) NLRP3IL1BPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023129987-A1 PYRIDAZINE DERIVATIVES AS MODULATORS OF NLRP3 INFLAMMASOME AND RELATED METHODS Neumora Therapeutics, Inc. (US) 2023-07-06 WO disclosed