SCHEMBL2580108

SCHEMBL2580108

CC(C)Oc1ccc2c(c1)CN(C(=O)O)CC2

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.49
HRH3 Q9Y5N1 2/20 0.48
HPGD P15428 1/20 0.48
S1PR1 P21453 4/20 0.47
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
ABHD6 Q9BV23 1/20 0.45
F10 P00742 5/20 0.45
PRSS1 P07477 4/20 0.45
PRSS2 P07478 4/20 0.45
PRSS3 P35030 4/20 0.45
PLG P00747 2/20 0.45
ACACB O00763 1/20 0.45
NR1H2 P55055 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753253 0.91 ACACB (0.46) ABCB1HRH3HPGDS1PR1ESR1
SCHEMBL5257657 0.88 ALDH1A1 (0.47) ABCB1HPGDS1PR1ESR1ESR2
SCHEMBL29098116 0.85 HPGD (0.49) HRH3HPGDS1PR1ESR1ESR2
SCHEMBL1265523 0.83 NR1H2 (0.67) ABCB1HRH3HPGDESR1ESR2
SCHEMBL27538580 0.80 HRH3 (0.52) HRH3HPGDESR1ESR2F10
SCHEMBL5137232 0.80 HRH3 (0.58) ABCB1HRH3HPGDABHD6F10
SCHEMBL30290475 0.80 HRH3 (0.52) HRH3S1PR1ESR1ESR2ABHD6
SCHEMBL11295872 0.79 ESR1 (0.71) ABCB1HPGDESR1ESR2ABHD6
SCHEMBL28533346 0.79 HRH3 (0.57) HRH3HPGDESR1ESR2F10
SCHEMBL29098077 0.78 GAA (0.50) ABCB1HRH3ESR1ESR2ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101346353-B Sulfonamide derivatives and their use in modulating metalloproteases SERONO LAB 2012-01-11 CN disclosed
EP-1951674-B1 SULFONAMIDE DERIVATIVES AND USE THEREOF FOR THE MODULATION OF METALLOPROTEINASES MERCK SERONO SA (CH) 2011-11-23 EP disclosed
CN-101346353-A Sulfonamide derivatives and their use in modulating metalloproteases SERONO LAB (CH) 2009-01-14 CN disclosed