SCHEMBL2580555

SCHEMBL2580555

N#CCCC(NC(=O)C1=NOC2(CCN(S(=O)(=O)c3cc(Cl)ccc3Cl)CC2)C1)C1CCCO1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.43
MEN1 O00255 1/20 0.43
ATM Q13315 1/20 0.38
POLB P06746 1/20 0.36
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 1/20 0.36
THRB P10828 1/20 0.36
CNR1 P21554 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 1/20 0.35
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RECQL P46063 1/20 0.34
ADRB2 P07550 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2402616 0.79 KMT2A (0.38) KMT2AMEN1ATMALDH1A1THRB
SCHEMBL2400757 0.78 KMT2A (0.47) KMT2AMEN1ATMPOLBALDH1A1
SCHEMBL2404636 0.75 ATM (0.43) KMT2AATMALDH1A1KDM4ECNR1
SCHEMBL6409831 0.74 ATM (0.55) KMT2AATMPOLBALDH1A1KDM4E
SCHEMBL6411053 0.72 KMT2A (0.46) KMT2AMEN1ATMPOLBALDH1A1
SCHEMBL2403568 0.71 NAMPT (0.42) KMT2AMEN1ATMALDH1A1CNR1
SCHEMBL2400090 0.70 CACNA1G (0.46) MAPTGAASMN1; SMN2ADRB2
SCHEMBL2400043 0.69 USP2 (0.42) KMT2AMEN1ATMALDH1A1CNR1
SCHEMBL2403236 0.68 ALDH1A1 (0.40) ATMPOLBALDH1A1TSHRNPSR1
SCHEMBL2400718 0.68 DRD4 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048890-B2 Analgesics; neuropathic pain; headaches; muscle relaxants; incontence; tinnitus; diarrhea; antiarrhythmia agents; antiischemic agents; antiinflammatory agents; antiulcer agents; antidepressants; antiepileptic agents GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed