SCHEMBL2581171

SCHEMBL2581171

Cc1ccc(S(=O)(=O)NC(Cc2ccccc2)C(=O)N2CCC3(CC2)CC(C(=O)NCCC#N)=NO3)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.49
HPN P05981 3/20 0.46
ST14 Q9Y5Y6 3/20 0.46
KMT2A Q03164 3/20 0.45
HGFAC Q04756 1/20 0.45
PLAU P00749 1/20 0.45
MMP9 P14780 1/20 0.43
CTSL P07711 2/20 0.43
F11 P03951 1/20 0.42
HTT P42858 1/20 0.42
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 2/20 0.42
MAPK1 P28482 1/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
POLB P06746 1/20 0.40
AIMP2 Q13155 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6409170 0.88 TP53 (0.47) TP53HPNST14KMT2AHGFAC
SCHEMBL6412715 0.88 TP53 (0.56) TP53HPNST14KMT2AHGFAC
SCHEMBL2403293 0.85 ALDH1A1 (0.48) TP53HPNST14KMT2AHGFAC
SCHEMBL6409811 0.81 TP53 (0.53) TP53HPNST14KMT2AHGFAC
SCHEMBL2401027 0.77 ALDH1A1 (0.48) ALDH1A1MAPK1
SCHEMBL6409841 0.75 TP53 (0.46) TP53HPNST14KMT2AHGFAC
SCHEMBL22500544 0.73 KMT2A (0.70) TP53HPNST14KMT2AHGFAC
SCHEMBL22500546 0.73 KMT2A (0.70) TP53HPNST14KMT2AHGFAC
SCHEMBL2579196 0.73 ALDH1A1 (0.45) KMT2ACTSLHTTALDH1A1MEN1
SCHEMBL2400743 0.72 ALDH1A1 (0.49) KMT2ACTSLHTTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048890-B2 Analgesics; neuropathic pain; headaches; muscle relaxants; incontence; tinnitus; diarrhea; antiarrhythmia agents; antiischemic agents; antiinflammatory agents; antiulcer agents; antidepressants; antiepileptic agents GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048890-B2 Analgesics; neuropathic pain; headaches; muscle relaxants; incontence; tinnitus; diarrhea; antiarrhythmia agents; antiischemic agents; antiinflammatory agents; antiulcer agents; antidepressants; antiepileptic agents GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed