SCHEMBL2581571

SCHEMBL2581571

C=C(C(=O)O)c1ccncc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.58
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 2/20 0.48
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 2/20 0.47
PLOD2 O00469 1/20 0.47
PLOD3 O60568 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
PLOD1 Q02809 1/20 0.47
HIF1A Q16665 1/20 0.47
KDM4E B2RXH2 2/20 0.45
MPO P05164 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CYP2A6 P11509 1/20 0.45
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7439433 0.98 NAPRT (0.56) NAPRTKMT2AMEN1ALDH1A1CYP1A2
Pyridine SCHEMBL28870562 0.85 KMT2A (0.52) NAPRTKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL12970081 0.83 NAPRT (0.50) NAPRTKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL713716 0.82 TSHR (0.47) NAPRTALDH1A1HPGDHTTHSD17B10
SCHEMBL2817706 0.79 NAPRT (0.50) NAPRTKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL10910929 0.79 NAPRT (0.50) NAPRTKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL28774639 0.79 NAPRT (0.50) NAPRTKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL44226 0.77 CES1 (0.52) NAPRTKMT2AMEN1ALDH1A1CYP3A4
Isonicotinic Acid SCHEMBL11898509 0.76 NAPRT (0.71) NAPRTKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL9419372 0.75 CES1 (0.50) NAPRTKMT2AMEN1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114591295-A Pyridine salt-containing N- (indoleacyl) -N' - (substituted) propyl hydrazide derivative, and preparation method and application thereof 贵州大学 2022-06-07 CN claimed
CN-103772576-B A kind of preparation method being applied to the sorbent material that pristinamycin is separated WANG JINMING (CN) 2016-03-09 CN claimed
CN-103772576-A Preparation method of adsorbing agent applied to pristinamycin separation WANG JINMING 2014-05-07 CN claimed
CN-114702506-B 11-carbonyl-20-ethoxy source oridonin and 14-OH esterified serial derivatives and application thereof 郑州大学 2023-08-22 CN disclosed
CN-110386919-B Nuclear transport modulators and uses thereof 卡尔约药物治疗公司 2023-07-14 CN disclosed
CN-110183422-B Nuclear transport modulators and uses thereof 卡尔约药物治疗公司 2023-07-14 CN disclosed
CN-113845557-B Tripterine pyridine acrylic acid derivative and preparation method and medical application thereof 中国药科大学 2022-07-22 CN disclosed
CN-114702506-A 11-carbonyl-20-ethoxy economic oridonin and 14-OH esterified series derivatives and application thereof 郑州大学 2022-07-05 CN disclosed
EP-3710439-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2020-09-23 EP disclosed
CN-110386919-A Nuclear translocation regulator and application thereof 卡尔约药物治疗公司 2019-10-29 CN disclosed
CN-110183422-A Nuclear translocation regulator and application thereof 卡尔约药物治疗公司 2019-08-30 CN disclosed
CN-1136213-C New benzothiophene, benzofuran and indole compounds, preparation method therefor and medicine composition containing same ɪά��ʵ���� 2004-01-28 CN disclosed
US-6444694-B1 ANTIPROLIFERATIVE AGENTS WYETH 2002-09-03 US disclosed
EP-0830345-B1 STYRYL BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PROD (US) 2001-09-05 EP disclosed
CN-1293192-A New benzothiophene, benzofuran and indole compounds, preparation method therefor and medicine composition containing same ADIR (FR) 2001-05-02 CN disclosed
EP-0830345-A1 STYRYL BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-25 EP disclosed
US-5612336-A Heterocyclic amide derivatives as tachykinin antagonists MERCK, SHARP & DOHME LTD. (GB) 1997-03-18 US disclosed
WO-1996039391-A1 STYRYL BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1996-12-12 WO disclosed
WO-1994001402-A1 HETEROCYCLIC AMIDE DERIVATIVES AS TACHYKININ DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-01-20 WO disclosed
EP-0074229-A1 Triazole gastric anti-secretory agents PFIZER INC. (US) 1983-03-16 EP disclosed