SCHEMBL25816162

SCHEMBL25816162

C=C(CCNC)NC(=O)COc1ccc2c(c1)OC(F)(F)O2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.43
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
SMYD3 Q9H7B4 1/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 3/20 0.36
GAA P10253 2/20 0.36
HPGD P15428 4/20 0.36
GLA P06280 1/20 0.36
CYP1A2 P05177 1/20 0.35
MAPT P10636 3/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
PKM P14618 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25801914 0.86 MRGPRX4 (0.46) MRGPRX4KMT2AMEN1ALDH1A1KDM4E
SCHEMBL20999307 0.85 MRGPRX4 (0.39) MRGPRX4KMT2AMEN1SMYD3ALDH1A1
SCHEMBL22956306 0.82 ADORA3 (0.42) MRGPRX4KMT2AMEN1HPGDCYP1A2
SCHEMBL22956371 0.79 MEN1 (0.39) MRGPRX4KMT2AMEN1ALDH1A1CYP1A2
SCHEMBL22628300 0.79 KMT2A (0.49) MRGPRX4KMT2AMEN1SMYD3CTNNB1
SCHEMBL22627759 0.79 KIT (0.47) MRGPRX4
SCHEMBL20999368 0.79 MRGPRX4 (0.35) MRGPRX4KMT2AMEN1ALDH1A1KDM4E
SCHEMBL22627932 0.78 BACE1 (0.35) MRGPRX4KMT2AMEN1SMYD3ALDH1A1
SCHEMBL22956329 0.78 GCGR (0.37) MRGPRX4KMT2ANPC1RAB9A
SCHEMBL25798610 0.78 SMN1; SMN2 (0.34) MRGPRX4KMT2AMEN1SMYD3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3452456-B1 BICYCLIC MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2023-07-05 EP disclosed