SCHEMBL2581743

SCHEMBL2581743

O=C(CCC(=O)ON1C(=O)C=CC1=O)ON1C(=O)C=CC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
HPGD P15428 4/20 0.41
BLM P54132 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
WRN Q14191 1/20 0.41
HIF1A Q16665 1/20 0.41
GSK3A P49840 2/20 0.39
GSK3B P49841 2/20 0.39
PTGS1 P23219 5/20 0.35
PTGS2 P35354 5/20 0.35
NSD2 O96028 1/20 0.33
G6PD P11413 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
MGLL Q99685 6/20 0.32
NPSR1 Q6W5P4 4/20 0.32
LMNA P02545 4/20 0.32
MAPT P10636 4/20 0.32
FAAH O00519 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28335153 0.92 PTGS1 (0.43) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL28390950 0.91 ALDH1A1 (0.38) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL17676438 0.90 ALDH1A1 (0.39) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL13356960 0.89 PTGS1 (0.44) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL15184862 0.89 ALDH1A1 (0.37) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL27885106 0.87 ALDH1A1 (0.36) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL714989 0.87 ALDH1A1 (0.44) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL269178 0.86 ALDH1A1 (0.41) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL5961226 0.86 PTGS1 (0.46) ALDH1A1HPGDBLMCYP1A2CYP2C19
SCHEMBL31121833 0.84 PTGS1 (0.49) ALDH1A1HPGDBLMCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115443134-A Conjugates of cell binding molecules and camptothecin analogs 杭州多禧生物科技有限公司 2022-12-06 CN disclosed
CN-113195487-A 2, 3-diaminosuccinyl conjugate linkers 杭州多禧生物科技有限公司 2021-07-30 CN disclosed
CN-112272669-A Cross-linked pyrrolobenzodiazepine dimer (PBD) derivatives and conjugates thereof 杭州多禧生物科技有限公司 2021-01-26 CN disclosed
CN-110621673-A Double-stranded linked cytotoxic drug conjugates 杭州多禧生物科技有限公司 2019-12-27 CN disclosed
EP-2384318-A2 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS Ardelyx, Inc. (US) 2011-11-09 EP disclosed
WO-2010078449-A2 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2010-07-08 WO disclosed