SCHEMBL25820506

SCHEMBL25820506

N#Cc1cc2c(=O)[nH]c(=O)[nH]c2c(F)c1Br

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPYD Q12882 1/20 0.38
IDH1 O75874 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
CSNK2A1 P68400 1/20 0.33
CHEK1 O14757 1/20 0.33
IDO1 P14902 5/20 0.31
FASN P49327 4/20 0.31
DAO P14920 1/20 0.30
PNP P00491 1/20 0.30
TYMP P19971 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25814975 0.79 IDH1 (0.39) IDH1CSNK2A2CSNK2BCSNK2A1PNP
SCHEMBL16637455 0.76 IDH1 (0.36) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL21379214 0.76 IDH1 (0.36) DPYDIDH1CSNK2A2CSNK2BCSNK2A1
SCHEMBL29592452 0.76 IDH1 (0.36) DPYDIDH1CSNK2A2CSNK2BCSNK2A1
SCHEMBL29388927 0.76 IDH1 (0.36) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL24004705 0.74 GRIN2D (0.38) IDH1CSNK2A2CSNK2BCSNK2A1PNP
SCHEMBL31542506 0.74 IDH1 (0.34) IDH1CSNK2A2CSNK2BCSNK2A1PNP
SCHEMBL25330088 0.72 SIRT2 (0.41) TYMP
SCHEMBL30504352 0.70 PGR (0.37) IDH1CSNK2A2CSNK2BCSNK2A1CHEK1
SCHEMBL22393852 0.70 PGR (0.37) IDH1CSNK2A2CSNK2BCSNK2A1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125989-A1 QUINAZOLINE COMPOUND AND APPLICATION THEREOF 上海医药集团股份有限公司 2023-07-06 WO disclosed