SCHEMBL25825900

SCHEMBL25825900

CCOC(=O)CC(=O)c1ccc2c(c1O)CN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.43
ESR2 Q92731 1/20 0.42
NR1H2 P55055 2/20 0.39
DDB1 Q16531 2/20 0.39
CRBN Q96SW2 2/20 0.39
NAMPT P43490 4/20 0.39
MIF P14174 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
ADORA1 P30542 1/20 0.36
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34
HSP90AA1 P07900 1/20 0.34
F13A1 P00488 1/20 0.34
TGM2 P21980 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25825838 0.83 ESR2 (0.35) HDAC1ESR2NR1H2NAMPTMIF
SCHEMBL25825899 0.81 ESR2 (0.49) HDAC1ESR2NR1H2DDB1CRBN
SCHEMBL25604140 0.81 HDAC1 (0.45) HDAC1ESR2NR1H2DDB1CRBN
SCHEMBL15893739 0.78 ESR2 (0.51) HDAC1ESR2NR1H2DDB1CRBN
SCHEMBL16269644 0.75 DDB1 (0.45) HDAC1ESR2NR1H2DDB1CRBN
SCHEMBL21496681 0.74 DDB1 (0.48) ESR2DDB1CRBNNAMPTMAPK1
SCHEMBL15896377 0.73 ESR2 (0.49) HDAC1ESR2NR1H2DDB1CRBN
SCHEMBL21805005 0.73 DDB1 (0.47) HDAC1ESR2NR1H2DDB1CRBN
SCHEMBL12682903 0.72 ADORA1 (0.53) ESR2NR1H2MAPK1ADORA1KMT2A
SCHEMBL15503203 0.71 ESR2 (0.56) HDAC1ESR2NR1H2NAMPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed