SCHEMBL2582641

SCHEMBL2582641

Cc1ccc(-c2ccc3c(c2)C2(C)CCNC(C3)[C@H]2C)nn1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.59
OPRD1 P41143 5/20 0.59
OPRK1 P41145 5/20 0.59
SIGMAR1 Q99720 5/20 0.59
MRGPRX2 Q96LB1 4/20 0.43
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
HSD11B1 P28845 1/20 0.33
P2RX7 Q99572 1/20 0.32
SLC22A1 O15245 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18408180 1.00 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1206692 1.00 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1207273 0.80 OPRM1 (0.60) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL18408074 0.80 OPRM1 (0.60) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL18407995 0.80 OPRD1 (0.63) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1207662 0.80 OPRD1 (0.63) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL18407971 0.80 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL18408225 0.80 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1207656 0.80 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1207890 0.80 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245014-B1 UREA DERIVATIVES OF BENZOMORPHANES AND RELATED SCAFFOLDS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE BOEHRINGER INGELHEIM INT (DE) 2011-11-02 EP disclosed