SCHEMBL25830809

SCHEMBL25830809

N#Cc1ccc(-c2ccc(C(F)(F)F)cc2)cc1-c1cc[nH]n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.43
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
AR P10275 6/20 0.40
PGR P06401 2/20 0.40
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
DGAT1 O75907 2/20 0.38
SOAT1 P35610 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM5A P29375 1/20 0.37
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
CNR1 P21554 1/20 0.36
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL25301898 0.99 KIF11 (0.42) KIF11CYP11B1CYP11B2ARPGR
Hydrochloric Acid SCHEMBL30510081 0.99 KIF11 (0.42) KIF11CYP11B1CYP11B2ARPGR
SCHEMBL25378423 0.85 CYP11B1 (0.47) CYP11B1CYP11B2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL25255925 0.84 CYP11B1 (0.46) CYP11B1CYP11B2ALDH1A1MAPT
SCHEMBL26192949 0.82 AR (0.46) CYP11B1CYP11B2ARPGRALDH1A1
SCHEMBL25378290 0.81 KIF11 (0.40) KIF11CYP11B1CYP11B2CTSSCTSK
SCHEMBL30510138 0.81 KIF11 (0.40) KIF11CYP11B1CYP11B2CTSSCTSK
SCHEMBL30509975 0.78 KDM5A (0.39) KIF11CYP11B1CYP11B2CTSSCTSK
SCHEMBL30510102 0.77 NPBWR1 (0.49) KIF11CYP11B1CYP11B2ARPGR
SCHEMBL25302186 0.77 NPBWR1 (0.49) KIF11CYP11B1CYP11B2ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023122780-A9 2-PYRAZOLE ANILINES AND RELATED ANALOGS FOR INHIBITING YAP/TAZ-TEAD THE KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO disclosed
WO-2023122780-A2 2-PYRAZOLE ANILINES AND RELATED ANALOGS FOR INHIBITING YAP/TAZ-TEAD THE KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-06-29 WO disclosed