SCHEMBL25833223

SCHEMBL25833223

CC(C)(C)OC(=O)N1CCC2(CCN(CC(=O)OCc3ccccc3)CC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
CYP2D6 P10635 5/20 0.49
USP2 O75604 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 1/20 0.49
MAPK1 P28482 1/20 0.49
OPRD1 P41143 1/20 0.48
OPRK1 P41145 1/20 0.48
CHRM2 P08172 2/20 0.47
CHRM3 P20309 2/20 0.47
CHRM4 P08173 1/20 0.47
CHRM1 P11229 1/20 0.47
TACR1 P25103 1/20 0.46
YAP1 P46937 1/20 0.44
HTT P42858 1/20 0.44
STS P08842 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30312809 0.92 MEN1 (0.51) MEN1KMT2ACYP2D6CYP3A4MAPK1
SCHEMBL14129449 0.90 CHRM2 (0.57) MEN1KMT2ACHRM2CHRM3CHRM4
SCHEMBL12004666 0.90 CHRM2 (0.57) MEN1KMT2ACHRM2CHRM3CHRM4
SCHEMBL7526966 0.90 CHRM2 (0.57) MEN1KMT2ACHRM2CHRM3CHRM4
SCHEMBL30121349 0.88 MEN1 (0.54) MEN1KMT2ACYP2D6USP2ALDH1A1
SCHEMBL25134189 0.86 CHRM2 (0.54) MEN1KMT2ACHRM2CHRM3CHRM4
SCHEMBL12526355 0.83 CYP2D6 (0.69) CYP2D6USP2ALDH1A1CYP3A4MAPK1
SCHEMBL14716132 0.83 ENPP2 (0.56) MEN1KMT2AUSP2CYP3A4OPRD1
SCHEMBL2629479 0.83 CYP11B2 (0.53) MEN1KMT2ACYP2D6ALDH1A1OPRD1
SCHEMBL2440617 0.83 ENPP2 (0.56) MEN1KMT2AUSP2CYP3A4OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125907-A1 DEGRADATION OF BRUTON'S TYROSINE KINASE (BTK) BY CONJUGATION OF BTK INHIBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE BEIGENE, LTD. (KY) 2023-07-06 WO disclosed