SCHEMBL25833432

SCHEMBL25833432

Cc1ccc(-c2ccc3nc(NC(=O)[C@@H]4C5C=CC(C5)[C@@H]4C(=O)O)sc3c2)cc1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.68
ABL1 P00519 10/20 0.55
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
PIK3CG P48736 2/20 0.53
POLB P06746 1/20 0.50
CASP6 P55212 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ITK Q08881 1/20 0.50
KIT P10721 2/20 0.49
PDGFRA P16234 2/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
DYRK1A Q13627 1/20 0.48
KCNK2 O95069 1/20 0.48
KCNK4 Q9NYG8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25260232 1.00 ALDH1A1 (0.68) ALDH1A1ABL1NPC1RAB9APIK3CG
SCHEMBL30450724 1.00 ALDH1A1 (0.68) ALDH1A1ABL1NPC1RAB9APIK3CG
SCHEMBL30450796 0.91 ALDH1A1 (0.74) ALDH1A1NPC1RAB9APOLBCASP6
SCHEMBL25260244 0.91 ALDH1A1 (0.74) ALDH1A1NPC1RAB9APOLBCASP6
SCHEMBL25832624 0.91 ALDH1A1 (0.74) ALDH1A1NPC1RAB9APOLBCASP6
SCHEMBL25259451 0.90 ALDH1A1 (0.66) ALDH1A1ABL1NPC1RAB9APIK3CG
SCHEMBL30450121 0.90 ALDH1A1 (0.66) ALDH1A1ABL1PIK3CGITKKIT
SCHEMBL25306737 0.90 ALDH1A1 (0.66) ALDH1A1ABL1PIK3CGITKKIT
SCHEMBL30450168 0.90 ALDH1A1 (0.66) ALDH1A1ABL1NPC1RAB9APIK3CG
SCHEMBL25833484 0.90 ALDH1A1 (0.66) ALDH1A1ABL1NPC1RAB9APIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131649-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-07-13 WO disclosed