SCHEMBL25834000

SCHEMBL25834000

CNC1(C)CCN(c2nccc(C#N)n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 1/20 0.47
RIPK1 Q13546 1/20 0.41
HTR1A P08908 4/20 0.38
CTSS P25774 3/20 0.38
CHRM2 P08172 1/20 0.38
ACACB O00763 3/20 0.37
CHRM4 P08173 1/20 0.36
PTPN11 Q06124 2/20 0.35
MAPK3 P27361 1/20 0.35
MAPK1 P28482 1/20 0.35
CTSK P43235 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22389879 0.84 PANK3 (0.50) PANK3RIPK1CTSSCHRM2ACACB
SCHEMBL28676196 0.78 RET (0.46) PANK3RIPK1CTSSCHRM2ACACB
SCHEMBL30004676 0.78 RET (0.46) PANK3RIPK1CTSSCHRM2ACACB
SCHEMBL31421020 0.78 PANK3 (0.49) PANK3RIPK1HTR1ACTSSACACB
SCHEMBL29324869 0.76 PANK3 (0.48) PANK3HTR1ACTSSACACBMAPK1
SCHEMBL28671204 0.75 PANK3 (0.47) PANK3RIPK1CTSSCHRM2ACACB
SCHEMBL30165199 0.74 ADRB1 (0.55) PANK3HTR1ACTSKKDM4EALDH1A1
SCHEMBL16432600 0.74 ADRB1 (0.55) PANK3HTR1ACTSKKDM4EALDH1A1
SCHEMBL10845137 0.74 ACHE (0.48) PANK3RIPK1HTR1ACTSSPTPN11
SCHEMBL567862 0.74 PIK3CA (0.50) PANK3ACACBMAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11696916-B2 Carboxamide-pyrimidine derivatives as SHP2 antagonists MERCK PATENT GMBH (DE) 2023-07-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11696916-B2 Carboxamide-pyrimidine derivatives as SHP2 antagonists PTPN5, PTPN2, PTPN1 PANK3 1328/4885RIPK1 447/4885HTR1A 4127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.