SCHEMBL2583651

SCHEMBL2583651

COc1ncnc2c1ncn2[C@@H]1O[C@H](CO)C[C@H]1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 3/20 0.52
ADORA3 P0DMS8 2/20 0.45
HIF1A Q16665 1/20 0.45
BCHE P06276 1/20 0.43
ADORA1 P30542 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
DPP4 P27487 1/20 0.43
MEN1 O00255 1/20 0.43
SLC28A1 O00337 1/20 0.43
MAP3K7 O43318 1/20 0.43
SLC28A2 O43868 1/20 0.43
GAPDH P04406 1/20 0.43
MAPK1 P28482 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
STAT6 P42226 1/20 0.43
PI4KA P42356 1/20 0.43
KMT2A Q03164 1/20 0.43
PI4K2B Q8TCG2 1/20 0.43
DOT1L Q8TEK3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2585394 1.00 SLC29A1 (0.52) SLC29A1ADORA3HIF1ABCHEADORA1
SCHEMBL12174032 1.00 SLC29A1 (0.52) SLC29A1ADORA3HIF1ABCHEADORA1
SCHEMBL23982354 1.00 SLC29A1 (0.52) SLC29A1ADORA3HIF1ABCHEADORA1
SCHEMBL23982564 1.00 SLC29A1 (0.52) SLC29A1ADORA3HIF1ABCHEADORA1
SCHEMBL12580037 0.88 SLC29A1 (0.43) SLC29A1BCHEADORA1SMN1; SMN2TP53
SCHEMBL8621079 0.88 SLC29A1 (0.43) SLC29A1BCHEADORA1SMN1; SMN2TP53
SCHEMBL21367453 0.88 SLC29A1 (0.43) SLC29A1BCHEADORA1SMN1; SMN2TP53
SCHEMBL8621084 0.88 SLC29A1 (0.43) SLC29A1BCHEADORA1SMN1; SMN2TP53
SCHEMBL3039007 0.85 SLC29A1 (0.55) SLC29A1ADORA3HIF1ABCHEADORA1
SCHEMBL2580979 0.84 CYP2C19 (0.47) SLC29A1ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10100076-B2 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation GILEAD PHARMASSET LLC (US) 2018-10-16 US disclosed
US-20140057863-A1 MODIFIED NUCLEOSIDES FOR THE TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION GILEAD SCIENCES, INC. (US) 2014-02-27 US disclosed
EP-2251015-B1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation GILEAD PHARMASSET LLC (US) 2013-02-20 EP disclosed
US-20110269707-A1 Modified nucleosides for the treatment of viral infections and abnormal cellullar proliferation PHARMASSET, INC. 2011-11-03 US disclosed
EP-2251015-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation Pharmasset, Inc. (US) 2010-11-17 EP disclosed
EP-1411954-A2 MODIFIED NUCLEOSIDES FOR TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION Pharmasset Limited (BB) 2004-04-28 EP disclosed
US-20030087873-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation PHARMASSET, INC. 2003-05-08 US disclosed
WO-2002032920-A2 MODIFIED NUCLEOSIDES FOR TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION PHARMASSET LIMITED (BB) 2002-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140057863-A1 MODIFIED NUCLEOSIDES FOR THE TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION SLC29A1, PNP, SLC29A2 SLC29A1 1/4885ADORA3 83/4885HIF1A 2226/4885
US-20110269707-A1 Modified nucleosides for the treatment of viral infections and abnormal cellullar proliferation PNP, ALPP, XDH SLC29A1 13/4885ADORA3 160/4885HIF1A 2633/4885
US-10100076-B2 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation SLC29A1, SLC29A2, PNP SLC29A1 1/4885ADORA3 61/4885HIF1A 2083/4885
US-20030087873-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation SLC29A1, PNP, SLC29A2 SLC29A1 1/4885ADORA3 82/4885HIF1A 2313/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.