SCHEMBL25838296

SCHEMBL25838296

Cc1cc2c(c([C@@H]3CCCN3)c1)CN(C(=O)c1ccnc(C)n1)CC2

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.35
CREBBP Q92793 1/20 0.33
PLA2G1B P04054 1/20 0.33
MAPT P10636 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
GAA P10253 1/20 0.32
SPR P35270 3/20 0.32
POLB P06746 1/20 0.32
BCL2 P10415 1/20 0.31
BAD Q92934 1/20 0.31
CFTR P13569 3/20 0.31
PDE2A O00408 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
BRD4 O60885 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
KDM2B Q8NHM5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25838305 0.88 KDM4E (0.38) PDE4BPLA2G1BMAPTATG4BSPR
SCHEMBL25838297 0.84 PDE4B (0.32) PDE4BPLA2G1BMAPTATG4BSPR
SCHEMBL25838291 0.84 HSP90AA1 (0.33) PDE4BPOLBHSP90AA1HSP90AB1
SCHEMBL25300385 0.82 MAP3K12 (0.36)
SCHEMBL30068705 0.82 MAP3K12 (0.36)
SCHEMBL25300384 0.82 MAP3K12 (0.36)
SCHEMBL25837869 0.81 PROKR1 (0.38) PDE4BMAPTMAPK1KDM2B
SCHEMBL25838318 0.80 SPR (0.35) SPRCFTRMAPK1HSP90AA1HSP90AB1
SCHEMBL25838322 0.79 HSP90AA1 (0.33) PDE4BMAPK1HSD17B10HSP90AA1HSP90AB1
SCHEMBL25837868 0.79 LMNA (0.36) PDE4BPOLBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed