SCHEMBL25838992

SCHEMBL25838992

CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc3c(c2)CCN(C(=O)OC(C)(C)C)C3)ncc1Cl

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AXL P30530 7/20 0.71
NEK2 P51955 1/20 0.59
AURKA O14965 1/20 0.57
AURKB Q96GD4 1/20 0.57
CCNK O75909 1/20 0.55
CCNA2 P20248 1/20 0.55
CDK2 P24941 1/20 0.55
CCND3 P30281 1/20 0.55
CDK9 P50750 1/20 0.55
CDK6 Q00534 1/20 0.55
ALK Q9UM73 10/20 0.52
MAP4K1 Q92918 1/20 0.50
INSR P06213 2/20 0.49
MET P08581 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30498941 1.00 AXL (0.71) AXLNEK2AURKAAURKBCCNK
SCHEMBL31173379 0.86 AXL (0.67) AXLNEK2AURKAAURKBALK
SCHEMBL25839123 0.86 AXL (0.67) AXLNEK2AURKAAURKBALK
SCHEMBL21446914 0.82 AXL (0.76) AXLNEK2AURKAAURKBCCNK
SCHEMBL31173432 0.82 AXL (0.74) AXLNEK2AURKAAURKBALK
SCHEMBL25837708 0.82 AXL (0.74) AXLNEK2AURKAAURKBALK
SCHEMBL31173541 0.81 AXL (0.76) AXLNEK2AURKAAURKBALK
SCHEMBL25837783 0.81 AXL (0.76) AXLNEK2AURKAAURKBALK
SCHEMBL31173443 0.81 AXL (0.75) AXLNEK2AURKAAURKBALK
SCHEMBL25837709 0.81 AXL (0.75) AXLNEK2AURKAAURKBALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134582-A1 PYRIMIDINE-2,4-DIAMINE DERIVATIVES AS WELL AS PREPARATION METHOD THEREFOR AND USE THEREOF 上海立森印迹医药技术有限公司 2023-07-20 WO disclosed