SCHEMBL25848883

SCHEMBL25848883

CS(=O)(=O)c1ccc(C(=O)NCc2ccc(Cl)cc2Cl)s1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
NLRP1 Q9C000 1/20 0.51
EPHX2 P34913 14/20 0.51
TSHR P16473 1/20 0.48
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30392482 1.00 LMNA (0.51) LMNAMAPK1NLRP1EPHX2TSHR
SCHEMBL25848762 0.89 HDAC1 (0.46) EPHX2HDAC1HDAC6
SCHEMBL25303214 0.89 LMNA (0.53) LMNAMAPK1NLRP1EPHX2TSHR
SCHEMBL25848879 0.88 EPHX2 (0.49) LMNAMAPK1NLRP1EPHX2TSHR
SCHEMBL30393345 0.88 EPHX2 (0.49) LMNAMAPK1NLRP1EPHX2TSHR
SCHEMBL25262922 0.84 EPHX2 (0.53) EPHX2
SCHEMBL25848789 0.79 HDAC1 (0.45) LMNAMAPK1NLRP1EPHX2HDAC1
SCHEMBL24196134 0.78 P2RX7 (0.43) EPHX2HDAC1HDAC6
SCHEMBL25848757 0.78 HDAC1 (0.44) LMNAMAPK1NLRP1EPHX2HDAC1
SCHEMBL25848904 0.78 EPHX2 (0.41) LMNAMAPK1NLRP1EPHX2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2023-07-13 US disclosed
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2023-07-13 US disclosed
CN-116075297-A KCNT1 inhibitors and methods of use 普拉西斯精密医药公司 2023-05-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE KCNT1, KCNT2, KCNQ2 LMNA 1423/4885MAPK1 890/4885NLRP1 3254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.