SCHEMBL2584929

SCHEMBL2584929

COc1ccc(Nc2nc(Nc3cccc(Cl)c3)nc3ccccc23)cc1

nearest known ligand 0.80

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 5/20 0.80
MERTK Q12866 5/20 0.67
SLC2A1 P11166 1/20 0.60
MAPT P10636 2/20 0.59
MAPK1 P28482 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
NPC1 O15118 1/20 0.59
ALDH1A1 P00352 1/20 0.59
TP53 P04637 1/20 0.59
RAB9A P51151 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
ABCG2 Q9UNQ0 3/20 0.57
PDE5A O76074 2/20 0.57
LMNA P02545 1/20 0.57
KDM4E B2RXH2 1/20 0.55
HTT P42858 1/20 0.55
TAAR1 Q96RJ0 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590759 0.89 NPY5R (0.76) NPY5RSLC2A1MAPTMAPK1MEN1
SCHEMBL8909187 0.89 NPY5R (1.00) NPY5RMERTKSLC2A1MAPTMAPK1
Hydrochloric Acid SCHEMBL8907334 0.88 NPY5R (0.83) NPY5RMERTKSLC2A1MAPTMAPK1
SCHEMBL2587936 0.88 NPY5R (0.84) NPY5RMAPTMEN1KMT2ANPC1
Hydrochloric Acid SCHEMBL8900478 0.88 NPY5R (0.97) NPY5RMERTKSLC2A1MAPTMAPK1
SCHEMBL2590796 0.88 NPY5R (0.97) NPY5RMERTKSLC2A1MAPTMAPK1
SCHEMBL2592190 0.87 NPY5R (0.78) NPY5RSLC2A1MAPTMAPK1MEN1
Hydrochloric Acid SCHEMBL8897702 0.87 NPY5R (0.94) NPY5RMERTKSLC2A1MAPTMAPK1
SCHEMBL2590586 0.86 SLC2A1 (0.73) NPY5RMERTKSLC2A1TP53PDE5A
SCHEMBL8891851 0.86 NPY5R (0.78) NPY5RMERTKMAPTMAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed