SCHEMBL2587936

SCHEMBL2587936

Clc1ccc(Nc2nc(Nc3cccc(Cl)c3)nc3ccccc23)cc1

nearest known ligand 0.84

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 7/20 0.84
PDE5A O76074 3/20 0.64
ABCG2 Q9UNQ0 2/20 0.64
SOS1 Q07889 1/20 0.60
KDM4E B2RXH2 3/20 0.59
EGFR P00533 2/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
FADS1 O60427 1/20 0.58
MEN1 O00255 1/20 0.58
ALDH1A1 P00352 1/20 0.58
MAPT P10636 1/20 0.58
HPGD P15428 1/20 0.58
ALOX12 P18054 1/20 0.58
KMT2A Q03164 1/20 0.58
TAAR1 Q96RJ0 1/20 0.58
LCK P06239 1/20 0.56
TP53 P04637 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590759 0.96 NPY5R (0.76) NPY5RPDE5AABCG2SOS1KDM4E
SCHEMBL8890555 0.92 NPY5R (1.00) NPY5RPDE5AABCG2KDM4ENPC1
SCHEMBL2592190 0.91 NPY5R (0.78) NPY5RPDE5AABCG2SOS1KDM4E
Hydrochloric Acid SCHEMBL8901136 0.90 NPY5R (0.97) NPY5RPDE5AABCG2KDM4ENPC1
SCHEMBL8892229 0.90 NPY5R (0.97) NPY5RPDE5AABCG2KDM4ENPC1
Hydrochloric Acid SCHEMBL8890165 0.89 NPY5R (0.94) NPY5RPDE5AABCG2KDM4ENPC1
SCHEMBL2584929 0.88 NPY5R (0.80) NPY5RPDE5AABCG2KDM4ENPC1
SCHEMBL2588890 0.84 SOS1 (0.70) NPY5RPDE5ASOS1KDM4EALDH1A1
SCHEMBL3581297 0.83 ULK1 (0.59) NPY5RPDE5AABCG2SOS1KDM4E
SCHEMBL2591063 0.83 NPY5R (1.00) NPY5RPDE5AABCG2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed