SCHEMBL25849490

SCHEMBL25849490

Cn1nnc2c(Br)cncc21

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 6/20 0.38
SLC9A1 P19634 1/20 0.35
KEAP1 Q14145 1/20 0.35
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24375535 0.78 SLC9A1 (0.36) SLC9A1KEAP1KDM4ELMNATSHR
SCHEMBL24499231 0.76 SLC9A1 (0.35) SLC9A1KEAP1KDM4ELMNATSHR
SCHEMBL21888877 0.73 KDM4E (0.34) SLC9A1KEAP1KDM4ELMNATSHR
SCHEMBL30929215 0.72 GRM2 (0.62) GRM2SLC9A1KEAP1
SCHEMBL19911637 0.72 GRM2 (0.62) GRM2SLC9A1KEAP1
SCHEMBL22425913 0.71 GRM2 (0.37) GRM2SLC9A1KEAP1KDM4ELMNA
SCHEMBL24944742 0.68 KDM4E (0.34) KDM4ETSHR
SCHEMBL22425950 0.67 GRM2 (0.37) GRM2SLC9A1KEAP1
SCHEMBL29442714 0.67 KEAP1 (0.38) GRM2SLC9A1KEAP1KDM4ELMNA
SCHEMBL31509642 0.67 ADORA2A (0.39) KDM4ELMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023132369-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND HAVING NRF2 ACTIVATION EFFECT 中外製薬株式会社 2023-07-13 WO disclosed