SCHEMBL25852502

SCHEMBL25852502

Cc1cc(C(C)CN(C)C)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
CCR5 P51681 1/20 0.35
PBK Q96KB5 3/20 0.35
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
AOC3 Q16853 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25853238 0.86 AKR1C3 (0.40) CCR5PBKHTR2AHRH1AOC3
SCHEMBL26901678 0.85 PDPK1 (0.39) CCR5HTR2AHRH1AOC3TDP1
SCHEMBL25852510 0.83 HTR2A (0.38) PBKHTR2AHRH1AOC3TDP1
SCHEMBL25833169 0.81 PARP1 (0.42) HTR2AHRH1AOC3TDP1
SCHEMBL25833224 0.81 AOC3 (0.33) PBKHTR2AHRH1AOC3TDP1
SCHEMBL8343177 0.79 ALDH1A1 (0.46) TSHRAKR1C3AKR1C2
SCHEMBL8281294 0.79 ALDH1A1 (0.46) TSHRAKR1C3AKR1C2
SCHEMBL20738580 0.78 ABCB11 (0.46) TSHRAKR1C3AKR1C2
SCHEMBL25857177 0.78 ABCB11 (0.46) TSHRAKR1C3AKR1C2
SCHEMBL5134118 0.76 HTR2A (0.38) TSHRHTR2AAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023135233-A1 AZAINDOLE DERIVATIVES AND THEIR USE AS ERK KINASE INHIBITORS AGV DISCOVERY (FR) 2023-07-20 WO disclosed