SCHEMBL25857423

SCHEMBL25857423

CNc1nc(C=O)cn2c1nc1ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.51
KDM4E B2RXH2 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ADORA2A P29274 13/20 0.42
ADORA1 P30542 9/20 0.42
HTR2C P28335 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
BRD4 O60885 1/20 0.38
H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 P62805 1/20 0.38
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
CRHBP P24387 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHR2 Q13324 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25308682 0.79 BRD4 (0.46) KDM4EADORA2AADORA1ALDH1A1GAA
SCHEMBL29435907 0.79 BRD4 (0.46) KDM4EADORA2AADORA1ALDH1A1GAA
SCHEMBL25306779 0.78 ADORA2A (0.58) ADORA2AADORA1
SCHEMBL25857612 0.76 TOP2A (0.52) TOP2AKDM4ESMN1; SMN2ADORA2AADORA1
SCHEMBL25858412 0.75 ADORA2A (0.64) TOP2AKDM4ESMN1; SMN2ADORA2AADORA1
SCHEMBL2816349 0.73 KDM4E (0.63) TOP2AKDM4ESMN1; SMN2ADORA2AADORA1
SCHEMBL29435897 0.71 ADORA2A (0.40) ADORA2AADORA1
SCHEMBL15722446 0.71 BRD4 (0.44) TOP2ABRD4H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16
SCHEMBL2820509 0.70 TOP2A (0.52) TOP2AKDM4ESMN1; SMN2ADORA2AADORA1
SCHEMBL2816600 0.70 TOP2A (0.52) TOP2AKDM4ESMN1; SMN2ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023130701-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF 中山大学 2023-07-13 WO disclosed