SCHEMBL25858412

SCHEMBL25858412

CNc1nc(CO)cn2c1nc1ccccc12

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.64
TOP2A P11388 1/20 0.51
ADORA1 P30542 11/20 0.48
HTR2C P28335 1/20 0.45
BRD4 O60885 1/20 0.43
H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 P62805 1/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
ADORA3 P0DMS8 2/20 0.41
ADORA2B P29275 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25857612 0.87 TOP2A (0.52) ADORA2ATOP2AADORA1HTR2CBRD4
SCHEMBL25857595 0.86 ADORA2A (0.64) ADORA2AADORA1KDM4EALDH1A1LMNA
SCHEMBL29435895 0.79 ADORA2A (0.52) ADORA2AADORA1BRD4
SCHEMBL25307292 0.79 ADORA2A (0.52) ADORA2AADORA1BRD4
SCHEMBL2820509 0.78 TOP2A (0.52) ADORA2ATOP2AADORA1HTR2CBRD4
SCHEMBL25857400 0.78 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL2816022 0.77 TOP2A (0.51) ADORA2ATOP2AADORA1HTR2CBRD4
SCHEMBL25857423 0.75 TOP2A (0.51) ADORA2ATOP2AADORA1HTR2CBRD4
SCHEMBL2816349 0.73 KDM4E (0.63) ADORA2ATOP2AADORA1HTR2CBRD4
SCHEMBL2816600 0.73 TOP2A (0.52) ADORA2ATOP2AADORA1HTR2CBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023165165-A1 BENZOIMIDAZOPYRAZINE-3-CARBOXAMIDE COMPOUND TARGETING A2A AND ANTI-TUMOR IMMUNOLOGICAL FUNCTION THEREOF 中山大学 2023-09-07 WO disclosed
WO-2023130701-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF 中山大学 2023-07-13 WO disclosed