SCHEMBL25857612

SCHEMBL25857612

CCc1cn2c(nc3ccccc32)c(NC)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.52
HTR2C P28335 1/20 0.52
ADORA2A P29274 6/20 0.49
ADORA1 P30542 4/20 0.49
BRD4 O60885 1/20 0.44
H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 P62805 1/20 0.44
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
TP53 P04637 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
HK1 P19367 1/20 0.40
HKDC1 Q2TB90 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25858412 0.87 ADORA2A (0.64) TOP2AHTR2CADORA2AADORA1BRD4
SCHEMBL2820509 0.80 TOP2A (0.52) TOP2AHTR2CADORA2AADORA1BRD4
SCHEMBL2816022 0.79 TOP2A (0.51) TOP2AHTR2CADORA2AADORA1BRD4
SCHEMBL25857423 0.76 TOP2A (0.51) TOP2AHTR2CADORA2AADORA1BRD4
SCHEMBL2816349 0.74 KDM4E (0.63) TOP2AHTR2CADORA2AADORA1BRD4
SCHEMBL25857595 0.73 ADORA2A (0.64) ADORA2AADORA1KDM4EALDH1A1HPGD
SCHEMBL2816603 0.71 KDM4E (0.53) TOP2AHTR2CADORA2AADORA1KDM4E
SCHEMBL2816600 0.71 TOP2A (0.52) TOP2AHTR2CADORA2AADORA1BRD4
SCHEMBL2820944 0.70 KDM4E (0.51) TOP2AHTR2CADORA2AADORA1KDM4E
SCHEMBL2816214 0.70 ADORA2A (0.63) TOP2AHTR2CADORA2AADORA1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023130701-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF 中山大学 2023-07-13 WO disclosed