SCHEMBL2586680

SCHEMBL2586680

COc1ccc(C(=O)N2CCc3oncc3C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.51
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
PDE4B Q07343 2/20 0.49
PDE4D Q08499 2/20 0.49
KMT2A Q03164 3/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
MEN1 O00255 2/20 0.47
POLB P06746 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HDAC6 Q9UBN7 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584773 0.77 HPGD (0.51) HPGDLMNAALDH1A1L3MBTL1
SCHEMBL8435113 0.77 HPGD (0.50) HPGDCA1CA2CA7CA9
SCHEMBL13302265 0.77 HPGD (0.69) HPGDCA1CA2CA7CA9
SCHEMBL30260147 0.77 HPGD (0.69) HPGDCA1CA2CA7CA9
SCHEMBL5524312 0.76 CA1 (0.72) HPGDCA1CA2CA7CA9
SCHEMBL5523403 0.76 CA1 (0.80) HPGDCA1CA2CA7CA9
SCHEMBL4259746 0.75 LMNA (0.50) HPGDMAPTLMNAPOLBALDH1A1
SCHEMBL20424296 0.74 MEN1 (0.35) HPGDPDE4BKMT2AMAPTLMNA
SCHEMBL5527334 0.74 HPGD (0.46) HPGDCA1CA2CA7CA9
SCHEMBL3052857 0.73 PDE4B (0.69) CA1CA2CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed