SCHEMBL2586781

SCHEMBL2586781

CC(C(=O)NO)(c1ccc(-c2noc(-c3cnn(-c4ccccc4)c3C(F)(F)F)n2)cc1)C1CCCCC1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 11/20 0.56
POLB P06746 2/20 0.39
DDR1 Q08345 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
DDR2 Q16832 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
MAP3K20 Q9NYL2 1/20 0.38
MAP3K2 Q9Y2U5 1/20 0.38
HDAC4 P56524 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CHUK O15111 1/20 0.38
TXNRD1 Q16881 1/20 0.38
NOX4 Q9NPH5 1/20 0.38
S1PR4 O95977 2/20 0.37
S1PR5 Q9H228 2/20 0.37
S1PR3 Q99500 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2586782 0.77 S1PR1 (0.54) S1PR1POLBHDAC4MAPTSMN1; SMN2
SCHEMBL2586779 0.77 S1PR1 (0.66) S1PR1S1PR4S1PR5S1PR3
SCHEMBL27903358 0.77 S1PR1 (0.64) S1PR1POLBHDAC4MAPTSMN1; SMN2
SCHEMBL12289131 0.76 S1PR1 (0.81) S1PR1POLBMAPTSMN1; SMN2
SCHEMBL2576403 0.75 S1PR1 (0.82) S1PR1POLBMAPTSMN1; SMN2
SCHEMBL27903357 0.75 S1PR1 (0.59) S1PR1POLBMAPTSMN1; SMN2CHUK
SCHEMBL2591289 0.74 S1PR1 (0.63) S1PR1POLBMAPTSMN1; SMN2CHUK
SCHEMBL27921152 0.73 S1PR1 (0.77) S1PR1POLBMAPTSMN1; SMN2CHUK
SCHEMBL2579544 0.73 S1PR1 (0.77) S1PR1POLBMAPTSMN1; SMN2CHUK
SCHEMBL14696286 0.73 S1PR1 (0.71) S1PR1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560969-A1 4 - (5 - ISOXAZOLYL OR 5 - PYRRAZOLYL -1,2,4- OXADIAZOL - 3 - YL) -MANDELIC ACID AMIDES AS SPHINGOSIN- 1 - PHOSPHATE 1 RRECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2013-02-27 EP disclosed
WO-2011133734-A1 4 - (5 - ISOXAZOLYL OR 5 - PYRRAZOLYL -1,2,4- OXADIAZOL - 3 - YL) -MANDELIC ACID AMIDES AS SPHINGOSIN- 1 - PHOSPHATE 1 RRECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-10-27 WO disclosed