SCHEMBL25869512

SCHEMBL25869512

NC(=O)[C@@H](N)Cc1ccc(Br)cn1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
PLAU P00749 1/20 0.39
TSHR P16473 2/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 2/20 0.36
FPR2 P25090 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
GBA1 P04062 1/20 0.35
FDPS P14324 1/20 0.34
CYP1A2 P05177 1/20 0.34
EPHX1 P07099 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4208145 0.87 CYP1A2 (0.47) ALDH1A1KDM4ETSHRRAB9ANPC1
SCHEMBL27729422 0.81 SIRT2 (0.44) ALDH1A1KDM4ETSHRRAB9ANPC1
SCHEMBL4214065 0.81 SIRT2 (0.44) ALDH1A1KDM4ETSHRRAB9ANPC1
Hydrochloric Acid SCHEMBL27729421 0.80 SIRT2 (0.43) ALDH1A1KDM4ETSHRRAB9ANPC1
Hydrochloric Acid SCHEMBL4219539 0.80 SIRT2 (0.43) ALDH1A1KDM4ETSHRRAB9ANPC1
SCHEMBL514259 0.75 ADRA2A (0.47) ALDH1A1KDM4EADRA2AADRA2BADRA2C
SCHEMBL23158732 0.74 GBA1 (0.41) ALDH1A1KDM4EADRA2AADRA2BADRA2C
SCHEMBL8121390 0.73 EPHX1 (0.50) KMT2AEPHX1
SCHEMBL21447170 0.73 EPHX1 (0.50) KMT2AEPHX1
SCHEMBL10250742 0.72 PTPRA (0.57) ALDH1A1TSHRRAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134656-A1 PEPTIDYL NITRILE COMPOUND AND USE THEREOF 上海壹典医药科技开发有限公司 2023-07-20 WO disclosed