SCHEMBL25870419

SCHEMBL25870419

CC(C)CC(=O)N1CCC2(CC1)CCN(c1ncc(NC(C)C)cn1)CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
CYP2D6 P10635 6/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 2/20 0.38
POLB P06746 1/20 0.38
HIF1A Q16665 1/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 2/20 0.37
RET P07949 1/20 0.37
PTPN1 P18031 1/20 0.37
PIK3R1 P27986 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25876321 0.81 CYP3A4 (0.43) CYP3A4MEN1KMT2AHSD17B10SMN1; SMN2
SCHEMBL25870687 0.79 CYP3A4 (0.41) CYP3A4MEN1KMT2AHSD17B10SMN1; SMN2
SCHEMBL25870421 0.77 ITGB3 (0.39) CYP3A4MEN1KMT2AALDH1A1HPGD
SCHEMBL27381769 0.75 POLB (0.55) CYP3A4MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL389894 0.70 KDM4E (0.56) MEN1KMT2AALDH1A1L3MBTL1POLB
SCHEMBL25589849 0.68 HRH4 (0.48) MEN1KMT2AHSD17B10ALDH1A1CYP1A2
SCHEMBL25870439 0.68 POLB (0.47) CYP3A4MEN1KMT2AALDH1A1CYP2D6
SCHEMBL24590204 0.67 POLB (0.49) CYP3A4KMT2ASMN1; SMN2ALDH1A1CYP2C9
SCHEMBL27425285 0.67 PTPN11 (0.44) ALDH1A1
SCHEMBL27381767 0.67 CYP2D6 (0.65) CYP3A4SMN1; SMN2ALDH1A1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116920-A1 PENTA- FUSED HEXA-HETEROCYCLIC COMPOUND, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE 杭州多域生物技术有限公司 2023-06-29 WO disclosed