SCHEMBL25870990

SCHEMBL25870990

C#CCNc1ccc(NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.50
PTPN11 Q06124 1/20 0.46
PSMB8 P28062 1/20 0.45
NAMPT P43490 1/20 0.45
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA9 Q16790 2/20 0.44
MAPT P10636 1/20 0.44
CA2 P00918 1/20 0.44
MAPKAPK2 P49137 3/20 0.42
DRD2 P14416 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
MAPK14 Q16539 1/20 0.42
MAP4K4 O95819 1/20 0.41
GLS O94925 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16946760 0.84 CYP17A1 (0.50) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL28098568 0.83 SMN1; SMN2 (0.56) CA12CA1CA9MAPTCA2
SCHEMBL4132208 0.83 CYP17A1 (0.56) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL13055402 0.83 CYP17A1 (0.59) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL30552299 0.82 NAMPT (0.53) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL5106835 0.82 CYP17A1 (0.54) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL433863 0.81 ELANE (0.44) CA12CA1CA9MAPTCA2
SCHEMBL254714 0.81 PTPN11 (0.51) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL13193491 0.81 CYP17A1 (0.52) CYP17A1PTPN11PSMB8NAMPTCA12
SCHEMBL18025366 0.81 CYP17A1 (0.47) CYP17A1PTPN11PSMB8NAMPTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134673-A1 HIGH-SELECTIVITY KCNQ4 POTASSIUM CHANNEL AGONIST, PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海药物研究所 2023-07-20 WO disclosed