SCHEMBL25871509

SCHEMBL25871509

Cc1cc(C#N)c(Br)c(F)c1N

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 3/20 0.35
ADRB2 P07550 3/20 0.34
ADRB1 P08588 1/20 0.34
ALDH1A1 P00352 4/20 0.33
TSHR P16473 2/20 0.33
KHK P50053 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 2/20 0.32
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
USP2 O75604 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
LMNA P02545 1/20 0.30
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9821000 0.85 EGLN2 (0.35) EGLN2ADRB2ADRB1ALDH1A1TSHR
SCHEMBL25871526 0.81 KHK (0.32) KHK
SCHEMBL25871524 0.79 XDH (0.40) ADRB2ADRB1KHK
SCHEMBL23948129 0.78 EGLN2 (0.37) EGLN2ADRB2ADRB1ALDH1A1TSHR
SCHEMBL22724579 0.77 ALDH1A1 (0.40) ALDH1A1TSHRTP53CYP3A4TDP1
SCHEMBL22063008 0.75 ALDH1A1 (0.39) ALDH1A1TSHRTP53CYP3A4TDP1
SCHEMBL31433854 0.75 ALDH1A1 (0.39) ALDH1A1TSHRTP53CYP3A4TDP1
Hydrochloric Acid SCHEMBL34461204 0.74 ALDH1A1 (0.37) ALDH1A1TSHRTP53CYP3A4TDP1
SCHEMBL21051816 0.72 KDM4E (0.40) EGLN2ALDH1A1TSHRCYP3A4KDM4E
SCHEMBL2656947 0.72 TSHR (0.36) EGLN2ADRB2ALDH1A1TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023137634-A1 TRICYCLIC COMPOUND, PREPARATION THEREFOR, PHARMACEUTICAL COMPOSITION AND USE 上海奕拓医药科技有限责任公司 2023-07-27 WO disclosed