SCHEMBL25877884

SCHEMBL25877884

Cc1ccc(OCCCC#N)cc1-c1ccnc(N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 5/20 0.42
AAK1 Q2M2I8 2/20 0.39
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
P2RY12 Q9H244 2/20 0.39
GSK3B P49841 2/20 0.39
REN P00797 1/20 0.37
ABL1 P00519 2/20 0.36
APP P05067 1/20 0.36
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PIM1 P11309 1/20 0.34
CDK9 P50750 1/20 0.34
DYRK2 Q92630 1/20 0.34
DYRK1B Q9Y463 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22272955 0.86 AAK1 (0.39) DYRK1AAAK1GSK3BRENABL1
SCHEMBL30091626 0.84 DYRK1A (0.44) DYRK1AAAK1GSK3BRENABL1
SCHEMBL22272939 0.84 DYRK1A (0.44) DYRK1AAAK1GSK3BRENABL1
SCHEMBL23927511 0.82 TSHR (0.46) DYRK1AAAK1GSK3BNPC1RAB9A
SCHEMBL30091686 0.82 TSHR (0.46) DYRK1AAAK1GSK3BNPC1RAB9A
SCHEMBL25877903 0.82 DYRK1A (0.49) DYRK1AAAK1GSK3BRENABL1
SCHEMBL22273007 0.81 DYRK1A (0.42) DYRK1AAAK1PDE3BPDE3AP2RY12
SCHEMBL23956537 0.80 DYRK1A (0.41) DYRK1AAAK1GSK3BRENABL1
SCHEMBL22272533 0.79 DYRK1A (0.43) DYRK1AAAK1GSK3BRENABL1
SCHEMBL22272613 0.79 DYRK1A (0.46) DYRK1AAAK1GSK3BRENPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138433-A2 AMIDE COMPOUND HAVING RIPK1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR, AND USE THEREOF 中国科学院上海药物研究所 2023-07-27 WO disclosed