SCHEMBL25877903

SCHEMBL25877903

COCCOc1ccc(C)c(-c2ccnc(N)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.49
MAOA P21397 1/20 0.44
GSK3B P49841 1/20 0.44
NOS3 P29474 2/20 0.41
NOS1 P29475 2/20 0.41
NOS2 P35228 2/20 0.41
CHEK2 O96017 2/20 0.40
AAK1 Q2M2I8 1/20 0.40
REN P00797 1/20 0.39
PIM1 P11309 1/20 0.39
CDK9 P50750 1/20 0.39
DYRK2 Q92630 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
ABL1 P00519 2/20 0.39
GRM4 Q14833 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
S1PR1 P21453 2/20 0.36
CHEK1 O14757 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22272613 0.96 DYRK1A (0.46) DYRK1AMAOAGSK3BNOS3NOS1
SCHEMBL22272533 0.86 DYRK1A (0.43) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL22272939 0.85 DYRK1A (0.44) DYRK1AMAOAGSK3BNOS3NOS1
SCHEMBL30091626 0.85 DYRK1A (0.44) DYRK1AMAOAGSK3BNOS3NOS1
SCHEMBL25877728 0.84 DYRK1A (0.64) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL23927511 0.84 TSHR (0.46) DYRK1AGSK3BAAK1KDM4E
SCHEMBL30091686 0.84 TSHR (0.46) DYRK1AGSK3BAAK1KDM4E
SCHEMBL22273007 0.82 DYRK1A (0.42) DYRK1AGSK3BAAK1
SCHEMBL25877884 0.82 DYRK1A (0.42) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL23956537 0.81 DYRK1A (0.41) DYRK1AMAOAGSK3BAAK1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138433-A2 AMIDE COMPOUND HAVING RIPK1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR, AND USE THEREOF 中国科学院上海药物研究所 2023-07-27 WO disclosed