SCHEMBL30091686

SCHEMBL30091686

CCCCCCCCOc1ccc(C)c(-c2ccnc(N)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
DYRK1A Q13627 2/20 0.43
PDE2A O00408 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
PTPN11 Q06124 3/20 0.40
GSK3B P49841 1/20 0.40
NR5A1 Q13285 1/20 0.40
DHFR P00374 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
PTPN1 P18031 1/20 0.39
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
AAK1 Q2M2I8 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23927511 1.00 TSHR (0.46) TSHRDYRK1APDE2ACYP3A4CYP2D6
SCHEMBL30091626 0.86 DYRK1A (0.44) DYRK1AGSK3BKDM4ENPC1RAB9A
SCHEMBL22272939 0.86 DYRK1A (0.44) DYRK1AGSK3BKDM4ENPC1RAB9A
SCHEMBL25877903 0.84 DYRK1A (0.49) DYRK1AGSK3BKDM4EAAK1
SCHEMBL25877884 0.82 DYRK1A (0.42) DYRK1AGSK3BNPC1RAB9AAAK1
SCHEMBL22273007 0.82 DYRK1A (0.42) DYRK1AGSK3BAAK1
SCHEMBL23956537 0.81 DYRK1A (0.41) DYRK1APDE2AGSK3BNPC1RAB9A
SCHEMBL22272613 0.81 DYRK1A (0.46) DYRK1AGSK3BKDM4EAAK1
SCHEMBL22272533 0.81 DYRK1A (0.43) DYRK1AGSK3BKDM4ENPC1RAB9A
SCHEMBL11612193 0.80 TSHR (0.58) TSHRNR5A1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166116-B Amido bridged heterocyclic compound, and composition and application thereof 北京赛特明强医药科技有限公司 2022-12-27 CN disclosed