SCHEMBL2589722

SCHEMBL2589722

COC(=O)C1CCCCC1c1nsc(C)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 1/20 0.43
CPT2 P23786 1/20 0.35
CPT1A P50416 1/20 0.35
CNR2 P34972 1/20 0.34
BDKRB1 P46663 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM3 P20309 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2596235 0.77 SLC6A2 (0.46) SLC6A2SLC6A4CPT2CPT1ACNR2
SCHEMBL2582981 0.74 FABP4 (0.37) ALDH1A1MEN1KMT2A
SCHEMBL2582985 0.74 FABP4 (0.37) ALDH1A1MEN1KMT2A
SCHEMBL16636099 0.73 SLC6A2 (0.45) SLC6A2SLC6A4CPT2CPT1ACNR2
SCHEMBL16635759 0.72 SLC6A2 (0.41) SLC6A2SLC6A4CPT2CPT1ACNR2
SCHEMBL2593261 0.69 CPT2 (0.48) SLC6A2SLC6A4CPT2CPT1ACHRM2
SCHEMBL13595131 0.68 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL11514730 0.68 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL272354 0.68 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL8058857 0.68 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569319-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-20 EP disclosed
WO-2011141396-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-17 WO disclosed