SCHEMBL2590300

SCHEMBL2590300

CC(C#N)CN=NC(C)(C)C#N

nearest known ligand 0.32

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8911469 1.00 TSHR (0.32) TSHR
SCHEMBL11809967 0.92 TSHR (0.32) TSHR
SCHEMBL15864178 0.85
SCHEMBL14893216 0.83 TRPA1 (0.31)
SCHEMBL2699502 0.83 TSHR (0.34) TSHR
SCHEMBL11203432 0.83 TRPA1 (0.31)
SCHEMBL6905189 0.83 TSHR (0.34) TSHR
SCHEMBL11357736 0.82
SCHEMBL9005197 0.79
SCHEMBL11364010 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629395-A THICKENERS SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1997-05-13 US claimed
EP-4460726-A1 NONLINEAR OPTICAL CHROMOPHORES HAVING SHORT-CHAIN BRIDGE STRUCTURES, LOW OPTICAL LOSS MATERIALS CONTAINING THE SAME, AND METHODS FOR PREPARING THE SAME Lightwave Logic, Inc. (US) 2024-11-13 EP disclosed
EP-4445212-A1 NONLINEAR OPTICAL CHROMOPHORES HAVING TETRAHYDROCARBAZOLE DONOR GROUPS, LYOTROPIC COMPOSITIONS CONTAINING THE SAME, AND METHODS OF POLING SUCH COMPOSITIONS Lightwave Logic, Inc. (US) 2024-10-16 EP disclosed
EP-4358968-A1 4-ETHYNYL-3-HYDROXY-TETRAHYDROFURANYL-ADENINE PHOSPHORAMIDATES AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS Rome Therapeutics, Inc. (US) 2024-05-01 EP disclosed
EP-4240738-A1 PYRAZOLE DERIVATIVES AS RET KINASE INHIBITORS Eli Lilly and Company (US) 2023-09-13 EP disclosed
WO-2023132934-A1 NONLINEAR OPTICAL CHROMOPHORES HAVING SHORT-CHAIN BRIDGE STRUCTURES, LOW OPTICAL LOSS MATERIALS CONTAINING THE SAME, AND METHODS FOR PREPARING THE SAME LIGHTWAVE LOGIC, INC. (US) 2023-07-13 WO disclosed
WO-2023107680-A1 NONLINEAR OPTICAL CHROMOPHORES HAVING TETRAHYDROCARBAZOLE DONOR GROUPS, LYOTROPIC COMPOSITIONS CONTAINING THE SAME, AND METHODS OF POLING SUCH COMPOSITIONS LIGHTWAVE LOGIC, INC. (US) 2023-06-15 WO disclosed
WO-2022098970-A9 PYRAZOLE DERIVATIVES AS RET KINASE INHIBITORS ELI LILLY AND COMPANY (US) 2023-04-27 WO disclosed
WO-2022271878-A1 4-ETHYNYL-3-HYDROXY-TETRAHYDROFURANYL-ADENINE PHOSPHORAMIDATES AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS ROME THERAPEUTICS, INC. (US) 2022-12-29 WO disclosed
EP-4100381-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2022-12-14 EP disclosed
US-4696983-A ANTIDEPOSIT AGENTS, CARBOXYL CONTAINING POLYMER AND SURFACTANT THE B. F. GOODRICH COMPANY (US) 1987-09-29 US disclosed
EP-0096392-A1 Novel aminoglycosides, process for production thereof and use thereof KOWA COMPANY, LTD. (JP) 1983-12-21 EP disclosed
EP-0033213-A2 Pigment dispersions containing copolymer pigment dispersants and methods of grinding pigment dispersions HÜLS AMERICA INC. (a Delaware corporation) (US) 1981-08-05 EP disclosed
US-4243789-A ACRYLATE, VINYLPYRROLIDONE THE B. F. GOODRICH COMPANY (US) 1981-01-06 US disclosed
US-4163097-A POLYETHERS CONTAINING MALEIMIDE GROUPS CIBA-GEIGY CORPORATION (US) 1979-07-31 US disclosed
US-4158731-A PHOTOSENSITIVE POLYAMIDES CONTAINING MALEIMIDE GROUPS CIBA-GEIGY CORPORATION (US) 1979-06-19 US disclosed
US-4158730-A CONTAINING PHOTOSENSITIVE MALEIMIDE GROUPS; PRINTING PLATES, RELIEF IMAGES CIBA-GEIGY CORPORATION (US) 1979-06-19 US disclosed
US-4145511-A CONTAINING N-VINYL-2-PYRROLIDONE, PREPOLYMER OF A POLYALKYLENE ETHER GLYCOL OR POLYESTER GLYCOL AND AN AROMATIC DIISOCYANATE THE B. F. GOODRICH COMPANY (US) 1979-03-20 US disclosed
US-4079041-A CONTAINING PHOTOSENSITIVE MALEIMIDO GROUPS, PHOTOCURABLE CIBA-GEIGY CORPORATION (US) 1978-03-14 US disclosed
US-4042388-A FREE RADICAL FORMERS, DYES CANON KABUSHIKI KAISHA (JA) 1977-08-16 US disclosed