SCHEMBL25905710

SCHEMBL25905710

COC(OC)c1c(F)cncc1CC(C)NC(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.37
CTSS P25774 3/20 0.37
AAK1 Q2M2I8 1/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA7 P43166 2/20 0.34
TRPA1 O75762 2/20 0.33
SCN9A Q15858 3/20 0.33
PTPN1 P18031 1/20 0.33
CA4 P22748 1/20 0.32
CA9 Q16790 1/20 0.32
ATM Q13315 1/20 0.32
SSTR3 P32745 1/20 0.32
SYK P43405 1/20 0.32
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25905691 0.78 CYP3A4 (0.36) AAK1CA1CA2CA7TRPA1
SCHEMBL26076630 0.74 DPP4 (0.46) CTSKCTSSAAK1CA1CA2
SCHEMBL5848976 0.74 CTSS (0.39) CTSKCTSSAAK1CA1CA2
SCHEMBL25908717 0.72 CTSS (0.43) CTSKCTSSAAK1CA1CA2
SCHEMBL22543040 0.72 CYP17A1 (0.39) AAK1SYK
SCHEMBL10074464 0.71 SCN9A (0.49) CTSKCTSSAAK1TRPA1SCN9A
SCHEMBL28535891 0.70 ACACB (0.43) CTSKCTSSCA1CA2CA7
SCHEMBL5756353 0.70 CTSS (0.36) CTSKCTSSAAK1CA1CA2
SCHEMBL25135359 0.68 IDO1 (0.35) AAK1
SCHEMBL13609238 0.67 HRH3 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024063576-A1 NOVEL QUINAZOLINE COMPOUND AS KRAS INHIBITOR 일동제약(주) 2024-03-28 WO disclosed
US-20230242552-A1 Nitrogen-Containing Heterocyclic Compound, Preparation Method Therefor and Use Thereof 280 Bio, Inc (US) 2023-08-03 US disclosed
US-20230242552-A1 Nitrogen-Containing Heterocyclic Compound, Preparation Method Therefor and Use Thereof 280 Bio, Inc (US) 2023-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242552-A1 Nitrogen-Containing Heterocyclic Compound, Preparation Method Therefor and Use Thereof NRAS, KRAS, RAB8A CTSK 4073/4885CTSS 2857/4885AAK1 3992/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.