SCHEMBL2590577

SCHEMBL2590577

CN1Cc2cc(C3(Cl)CCC(c4nsc5cccnc45)CC3)ccc2-n2cnnc2C1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 4/20 0.32
AVPR2 P30518 2/20 0.32
KCNH2 Q12809 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2579842 0.86 AVPR1A (0.31) AVPR1A
SCHEMBL2586788 0.85 OXTR (0.32) AVPR1AAVPR2KCNH2
SCHEMBL2563008 0.84 AVPR1A (0.36) AVPR1AAVPR2KCNH2
SCHEMBL2563323 0.78 AVPR1A (0.33) AVPR1A
SCHEMBL2561816 0.77 AVPR1A (0.36) AVPR1AAVPR2KCNH2
SCHEMBL2563133 0.77 CBLB (0.32) AVPR1A
SCHEMBL2552411 0.77 AVPR1A (0.34) AVPR1AKCNH2
SCHEMBL2475282 0.76 AVPR1A (0.38) AVPR1AAVPR2KCNH2
SCHEMBL2560012 0.76 AVPR1A (0.32) AVPR1AAVPR2KCNH2
SCHEMBL2346991 0.76 SLC6A4 (0.32) AVPR1AAVPR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571879-A1 HETEROBIARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-27 EP claimed
WO-2011134877-A1 HETEROBIARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-03 WO claimed