SCHEMBL2552411

SCHEMBL2552411

CN1Cc2cc(C3(Cl)CCC(c4ccc(F)cc4)CC3)ccc2-n2cnnc2C1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 5/20 0.34
TACR1 P25103 3/20 0.34
SLC6A4 P31645 3/20 0.34
KCNH2 Q12809 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2549529 0.85 AVPR2 (0.35) AVPR1ATACR1KCNH2
SCHEMBL2563008 0.84 AVPR1A (0.36) AVPR1AKCNH2
Hydrochloric Acid SCHEMBL2544777 0.83 AVPR1A (0.33) AVPR1A
SCHEMBL2346991 0.82 SLC6A4 (0.32) AVPR1ASLC6A4KCNH2
SCHEMBL2472145 0.81 AVPR2 (0.34) AVPR1AKCNH2
SCHEMBL2336166 0.81 AVPR1A (0.31) AVPR1AKCNH2
SCHEMBL2563323 0.81 AVPR1A (0.33) AVPR1A
SCHEMBL2341614 0.80 AVPR2 (0.32) AVPR1AKCNH2
SCHEMBL2339933 0.80 IDH1 (0.31) AVPR1AKCNH2
SCHEMBL2556595 0.80 CYP11B2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011120877-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-06 WO disclosed