SCHEMBL2590769

SCHEMBL2590769

Clc1ccc2nc(NCc3ccccc3)nc(NCc3ccccc3)c2c1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.68
KDM4E B2RXH2 1/20 0.66
ALDH1A1 P00352 1/20 0.66
LMNA P02545 1/20 0.66
MAPT P10636 1/20 0.66
PKM P14618 1/20 0.66
UBE2N P61088 1/20 0.66
KMT2A Q03164 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
RCE1 Q9Y256 1/20 0.66
PDE5A O76074 5/20 0.62
HTR3A P46098 1/20 0.61
HRH4 Q9H3N8 1/20 0.61
APP P05067 7/20 0.59
BCHE P06276 4/20 0.59
ACHE P22303 4/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16280680 0.90 BCHE (0.57) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL2587220 0.90 RAD52 (0.70) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL3638867 0.88 PDE5A (0.73) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL2590671 0.85 RAD52 (0.82) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL2587383 0.85 RAD52 (0.76) RAD52KDM4EALDH1A1LMNAMAPT
Hydrochloric Acid SCHEMBL3636898 0.84 KDM4E (0.83) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL16280938 0.84 RAD52 (0.79) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL2591004 0.82 RAD52 (0.68) RAD52KDM4EALDH1A1LMNAMAPT
SCHEMBL9921364 0.81 LMNA (0.72) KDM4EALDH1A1LMNAMAPTKMT2A
SCHEMBL12175837 0.81 RAD52 (1.00) RAD52KDM4EALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed