SCHEMBL2590788

SCHEMBL2590788

Cc1c(P(=O)(c2ccccc2)c2ccccc2)c2ccccc2n1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 6/20 1.00
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
GLA P06280 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.47
MAPT P10636 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
GPR3 P46089 1/20 0.45
PGR P06401 1/20 0.42
NQO2 P16083 1/20 0.42
ALKBH5 Q6P6C2 1/20 0.40
FTO Q9C0B1 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29362654 1.00 NPSR1 (1.00) NPSR1KDM4EALDH1A1GAAHPGD
SCHEMBL2595693 0.81 NPSR1 (1.00) NPSR1KDM4EALDH1A1GAAHPGD
SCHEMBL17589451 0.72 NPSR1 (0.55) NPSR1ALDH1A1GAAHTTMAPT
SCHEMBL11991061 0.71 NPSR1 (0.53) NPSR1ALDH1A1GAAHTTMAPT
SCHEMBL14076803 0.70 NPSR1 (0.54) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL14020807 0.70 CA2 (0.52) NPSR1ALDH1A1GAAHTTMAPT
SCHEMBL17403754 0.69 NPSR1 (0.52) NPSR1ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL12175523 0.69 NPSR1 (0.68) NPSR1KDM4EALDH1A1HPGDHTT
SCHEMBL22379230 0.69 NPSR1 (0.53) NPSR1KDM4EALDH1A1GAAHSD17B10
SCHEMBL31132408 0.69 GPR3 (0.61) NPSR1KDM4EALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113980049-A Preparation method of diphenylphosphine substituted indole derivative 河南省科学院化学研究所有限公司 2022-01-28 CN disclosed
WO-2011137220-A1 SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-11-03 WO disclosed
WO-2011137220-A1 SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-11-03 WO disclosed