SCHEMBL2590838

SCHEMBL2590838

O=C1C=CNNC1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10915 0.73
SCHEMBL4113248 0.73
Hydrogen Sulfide SCHEMBL27545450 0.71
Hydrochloric Acid SCHEMBL17363299 0.71
SCHEMBL6223914 0.67
Pyrrolidine SCHEMBL15346082 0.62 ALDH1A1 (0.35)
SCHEMBL17912372 0.61
Piperidine SCHEMBL15346185 0.61 ALDH1A1 (0.39)
SCHEMBL9525717 0.59
SCHEMBL723377 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566864-A2 PYRIDAZINONES AS GPR119 AGONISTS Boehringer Ingelheim International GmbH (DE) 2013-03-13 EP claimed
WO-2011138427-A2 PYRIDAZINONES AS GPR119 AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-10 WO claimed
CN-1071090-C composition with synergistic fungicidal action ROHM & HAAS (US) 2001-09-19 CN claimed
CN-1189293-A Pyridazinones as marine antifouling agents ROHM & HAAS (US) 1998-08-05 CN claimed
CN-1038249-C Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM & HAAS (US) 1998-05-06 CN claimed
CN-1146282-A Composition with synergistic mycotoxicity effect ROHM & HAAS (US) 1997-04-02 CN claimed
CN-1069729-A Dihydropyridazinone, pyridazinone and related compound thereof as sterilant ROHM & HAAS (US) 1993-03-10 CN claimed
EP-0515257-A1 1-phenyl-1,4-dihydro-3-hydroxy-4-oxo-pyridazine derivatives, their preparation and their therapeutic use PIERRE FABRE MEDICAMENT (FR) 1992-11-25 EP claimed
EP-0175363-B1 4,5-DIHYDRO-3(2H)-PYRIDAZINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE CASSELLA Aktiengesellschaft (DE) 1990-01-17 EP claimed
CN-117460723-A Pharmaceutical compounds 杜克街生物有限公司 2024-01-26 CN disclosed
CN-115003296-A Compounds and methods for treating cystic fibrosis 弗拉特利发现实验室有限责任公司 2022-09-02 CN disclosed
CN-113646050-A Thieno [3,2-B ] pyrrolo [3,2-D ] pyridazinone derivatives and their use as PKM2 derivatives for the treatment of cancer, obesity and diabetes related disorders 安吉奥斯医药品有限公司 2021-11-12 CN disclosed
CN-103690542-B Poly-(ADP-ribose) AG14361 ABBVIE INC. (US) 2015-11-18 CN disclosed
CN-103690542-A Inhibitors of poly(ADP-ribose)polymerase ABBVIE INC 2014-04-02 CN disclosed
CN-1071090-C composition with synergistic fungicidal action ROHM & HAAS (US) 2001-09-19 CN disclosed
CN-1038249-C Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM & HAAS (US) 1998-05-06 CN disclosed
CN-1146282-A Composition with synergistic mycotoxicity effect ROHM & HAAS (US) 1997-04-02 CN disclosed
CN-1143637-A Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides ROHM & HAAS (US) 1997-02-26 CN disclosed
CN-1069729-A Dihydropyridazinone, pyridazinone and related compound thereof as sterilant ROHM & HAAS (US) 1993-03-10 CN disclosed
EP-0515257-A1 1-phenyl-1,4-dihydro-3-hydroxy-4-oxo-pyridazine derivatives, their preparation and their therapeutic use PIERRE FABRE MEDICAMENT (FR) 1992-11-25 EP disclosed