SCHEMBL25908428

SCHEMBL25908428

FC(F)(F)COc1cc(N2C[C@@H]3C[C@H]2CO3)nc2ccnn12

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 16/20 0.44
MAP3K13 O43283 2/20 0.43
PIK3R1 P27986 3/20 0.39
PIK3CA P42336 3/20 0.39
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25908430 1.00 MAP3K12 (0.44) MAP3K12MAP3K13PIK3R1PIK3CASYK
SCHEMBL25908431 0.77 PIK3CA (0.42) MAP3K12PIK3CA
SCHEMBL25908367 0.77 PIK3CA (0.36) MAP3K12PIK3R1PIK3CA
SCHEMBL25908374 0.71 KCNN3 (0.35)
SCHEMBL25908373 0.70 PDE10A (0.51)
SCHEMBL25908694 0.69 MAP3K7 (0.45) MAP3K12MAP3K13PIK3R1PIK3CA
SCHEMBL31674973 0.66 MAP3K12 (0.55) MAP3K12MAP3K13PIK3R1PIK3CA
SCHEMBL16224347 0.66 MAP3K12 (0.55) MAP3K12MAP3K13PIK3R1PIK3CA
SCHEMBL18307182 0.64 MAP3K12 (0.48) MAP3K12MAP3K13
SCHEMBL18307132 0.64 MAP3K12 (0.48) MAP3K12MAP3K13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138343-A1 NEW TYPE PYRAZOLOPYRIMIDINE COMPOUND AND COMPOSITION THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF 江苏亚尧生物科技有限公司 2023-07-27 WO disclosed