SCHEMBL2592358

SCHEMBL2592358

COc1c(C=O)[nH]c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
KDM4E B2RXH2 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
MAPK1 P28482 1/20 0.43
NR4A2 P43354 2/20 0.42
MCL1 Q07820 1/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
RAB9A P51151 1/20 0.42
KIF11 P52732 2/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
ABCG2 Q9UNQ0 3/20 0.41
ALOX15 P16050 1/20 0.41
ERN1 O75460 1/20 0.41
TUBB4A P04350 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15759926 0.80 KMT2A (0.61) ALDH1A1KDM4ENR4A2MAPTKMT2A
SCHEMBL29956558 0.76 AHR (0.55) ALDH1A1KDM4ESMN1; SMN2NR4A2MEN1
SCHEMBL1254486 0.76 AHR (0.55) ALDH1A1KDM4ESMN1; SMN2NR4A2MEN1
SCHEMBL4065612 0.74 KDM4E (0.72) ALDH1A1KDM4ESMN1; SMN2MAPK1MEN1
SCHEMBL5917605 0.73 NR4A2 (0.69) ALDH1A1KDM4ENR4A2MEN1KMT2A
SCHEMBL670200 0.73 AHR (0.57) ALDH1A1KDM4ESMN1; SMN2MAPK1NR4A2
SCHEMBL28136136 0.73 AHR (0.49) ALDH1A1KDM4ESMN1; SMN2MEN1MAPT
SCHEMBL4208427 0.73 KDM4E (0.51) ALDH1A1KDM4ESMN1; SMN2MAPK1NR4A2
SCHEMBL7311550 0.72 KDM4E (0.44) ALDH1A1KDM4ESMN1; SMN2MAPK1NR4A2
SCHEMBL1163942 0.72 MAPT (0.55) ALDH1A1KDM4ESMN1; SMN2MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011139242-A2 PROCESS FOR THE PREPARATION OF 2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLE DERIVATIVES USTAV EXPIREMENTÁLNEJ FARMAKOLÓGIE A TOXIKOLÓGIE SAV (SK) 2011-11-10 WO disclosed