SCHEMBL2592508

SCHEMBL2592508

Cc1c(-c2ccco2)n[nH]c1-c1ccc(N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.51
ADORA2A P29274 5/20 0.43
ADORA1 P30542 4/20 0.43
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PDE10A Q9Y233 1/20 0.41
PDPK1 O15530 1/20 0.41
HSD17B10 Q99714 7/20 0.40
ALDH1A1 P00352 7/20 0.40
KDM4E B2RXH2 6/20 0.40
HPGD P15428 4/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
MAPT P10636 3/20 0.40
MEN1 O00255 3/20 0.40
CASP1 P29466 3/20 0.40
BLM P54132 3/20 0.40
KMT2A Q03164 3/20 0.40
USP2 O75604 2/20 0.40
POLB P06746 2/20 0.40
PKM P14618 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1701229 0.84 PDPK1 (0.40) TAAR1ADORA2AADORA1HSP90AA1HSP90AB1
SCHEMBL10305768 0.79 ADORA2A (0.49) ADORA2AADORA1HSP90AA1HSP90AB1PDE10A
SCHEMBL2591881 0.72 MAPT (0.45) PDE10AHSD17B10ALDH1A1KDM4EHPGD
SCHEMBL2592615 0.72 HSP90AA1 (0.35) ADORA2AADORA1HSP90AA1HSP90AB1PDE10A
SCHEMBL1161258 0.70 TAAR1 (1.00) TAAR1ADORA2AHSD17B10ALDH1A1KDM4E
SCHEMBL1701209 0.69 HSP90AA1 (0.48) ADORA2AADORA1HSP90AA1HSP90AB1PDE10A
SCHEMBL27203335 0.69 MAPT (0.43) ADORA2AADORA1HSP90AA1HSP90AB1PDE10A
SCHEMBL27512201 0.68 KDM4E (0.50) ADORA2AADORA1HSP90AA1HSP90AB1PDE10A
SCHEMBL26905277 0.68 MAPT (0.52) HSP90AA1HSP90AB1PDE10AHSD17B10ALDH1A1
SCHEMBL5257770 0.66 CHEK1 (0.49) PDE10APDPK1HSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563759-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-03-06 EP disclosed
WO-2011139765-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2011-11-10 WO disclosed